Tamoxifen 10mg@30Tabs by Sopharma THE BEST STUFF
Pharmaceutical Name: Tamoxifen Citrate
Average Dose: 10-30 mg / day
Tamoxifen (Nolvadex, Nolvaxyl) is a subsequent cycle of steroids. The active ingredient is tamoxifen citrate.
Tamoxifen citrate is probably the most popular drug for aids male steroid users who want to avoid the effects estrogen? The use of anabolic steroids. Tamoxifen citrate binds to the estrogen receptor that blocks the action of hormones on target tissues and the achievement of an anti-estrogen.
Tamoxifen citrate is a selective modulator of estrogen receptor. Selective modulators of estrogen receptor can act as estrogen receptor agonists or antagonists. This activity of tamoxifen citrate is tissue selective, affecting estrogen receptors in the liver, breast, and? Bone. When the molecule of tamoxifen binds to this receptor, estrogen is blocked and can not have any influence, which in this tissue remaining inactive. Thus, an “anti-estrogenic” effect is achieved. The drug was developed and is still used to treat breast cancer. It is often used as first choice because of its mild compared with aromatase inhibitors. Of course you want to use the compound as smooth as possible when it comes to estrogen levels in women, but one could afford to be more aggressive in dealing with male strength athletes or bodybuilders.
As for its use in steroid users, Nolvaxyl can help in two ways. First, because the affinity of the compound that is capable of assisting in the prevention of gynecomastia. Tamoxifen citrate will compete with estrogen for estrogen receptors in some tissues, including breast, and If it can bind to estrogen receptors not have the opportunity to interact with the receptor and therefore the gynecomastia should not be able to develop. When the use of anabolic steroids can be converted to estradiol (estrogen) this protection against gynecomastia can be very valuable. However, it should be noted that tamoxifen citrate not eliminate the estrogen or not allow conversion to occur. Instead, attempts to counteract the effects of estrogen circulating in the body tissues the effects of drugs. Therefore, there is no evidence that the effects Nolvadex counteract the side effects are not related etrogenic tissues that are not in the breast, liver or bones. That is, there is no real causal connection to any reduction in water retention and acne on users who start taking tamoxifen citrate in relation to estrogen.